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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T39727 | ERα degrader-2 | ERK | |
ERα degrader-2 is a selective and potent estrogen receptor (SERD) degrader with anticancer activity, inhibits ERα, and has an EC50 value for estrogen receptor degradation of 0.3 nM.ERα degrader-2 can be used for the prev... | |||
T18605 | PROTAC ERα Degrader-2 | Others | |
PROTAC ERα Degrader-2 is composed of a cIAP1 ligand binding group, a linker, and an estrogen receptor α (ERα) binding group, serving as an ERα degrader. It achieves maximal ERα degradation in human mammary tumor MCF7 cel... |